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副研究员

杨亚军

职 称:副研究员

所属科室:合成药物化学研究室

导师类别:硕士生导师

联系方式:yangyajun@www.myhortonhome.com

所属重点实验室:活性物质发现与适药化研究北京市重点实验室

个人简介

教育背景:
2005/9 - 2010/7 北京协和医学院,药物化学,博士
2001/9 - 2005/7 河北医科大学,药学,学士
工作经历:
2014/5 - 至今 中国医学科学院,bobapp官方中国有限公司 ,副研究员
2010/7 - 2014/5 中国医学科学院,医学实验动物bobapp官方下载 ,助理研究员

研究方向

1、 新药先导化合物的发现与优化
2、 活性天然产物的合成与结构改造

发表论文

1. Yajun Yang, Jiangning Liu*, Xiandao Pan*. Synthesis and antiviral activity of lycorine derivatives. Journal of Asian Natural Products Research, 2020, 22(12): 1188-1196.
2. Yajun Yang, Ke Wang, Bo Wu, Ying Yang, Fangfang Lai, Xiaoguang Chen, Zhiyan Xiao*. Design, synthesis and biological evaluation of triaryl compounds as novel 20S proteasome inhibitors. Bioorg Med Chem Lett, 2020, 30(21):127508.
3. Shuo Pang, Caixian Sun, Shang Gao, Yajun Yang*, Xiandao Pan*, Lianfeng Zhang*. Evodiamine derivatives improve cognitive abilities in APPswe/ PS1ΔE9 transgenic mouse models of Alzheimer's disease. Animal Models and Experimental Medicine, 2020, 3(3):193-199.
4. Yajun Yang, Cuiju Zhu, Min Zhang, Shijun Huang, Jingjing Lin, Xiandao Pan*, Weiping Su*. Condensation of anthranilic acids with pyridines to furnish pyridoquinazolones via pyridine dearomatization. Chem Comm, 2016, 52(87): 12869-12872. .
5. Yajun Yang, Feifei Guan, Ling Bai, Li Zhang, Jiangning Liu, Xiandao Pan*, Lianfeng Zhang*. Quinolizidine alkaloids reduced mortality in EV71-infected mice by compensating for the levels of T cells. Bioorg Med Chem Lett, 2015, 35(17): 3526-3528.
6. Yajun Yang, Jing Ma, Jinghui Xiu, Ling Bai, Feifei Guan, Li Zhang, Jiangning Liu, Lianfeng Zhang*. Deferoxamine Compensates for Decreases in B Cell Counts and Reduces Mortality in Enterovirus 71-Infected Mice. Mar. Drugs, 2014, 12, 4086-4095.
7. Yajun Yang, Jinghui Xiu, Jiangning Liu, Li Zhang, Xiaoying Li, Yanfeng Xu, Chuan Qin, Lianfeng Zhang*. Chebulagic acid, a hydrolyzable tannin, exhibited antiviral activity in vitro and in vivo against human enterovirus 71. International Journal of Molecular Science, 2013, 14(5): 9618-9627.
8. Yajun Yang, Jinghui Xiu, Lianfeng Zhang, Chuan Qin, Jiangning Liu*. Antiviral activity of punicalagin toward human enterovirus 71 in vitro and in vivo. Phytomedicine, 2012, 20(1): 67-70.
9. Yajun Yang, Lianfeng Zhang, XiaoXu Fan, Chuan Qin, Jiangning Liu*. Antiviral effect of geraniin on human enterovirus 71 in vitro and in vivo. Bioorg Med Chem Lett, 2012, 22(6):2209-2211.
10. Yajun Yang, Yanan Yang, Jianshuang Jiang, Ziming Feng, Hongyan Liu, Xiandao Pan, Peicheng Zhang*. Synthesis and cytotoxic activity of heterocyclic ring-substituted phthalimide derivatives. Chin Chem Lett, 2010, 21(8): 902-904.

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